茶碱

分析标准品,HPLC≥98%

Theophylline

CAS号：58-55-9

分子式：C7H8N4O2

分子量：180.16

MDL：MFCD00079619

别名：1,3-二甲基黄嘌呤;2,6-二氧-1,3-二甲基嘌呤;3,7-二氢-1,3-二甲基-1H-嘌呤-2,6-二酮;2,6-二羟基-1,3-二甲基嘌呤

产品介绍

 Theophylline (1,3-Dimethylxanthine) 是有效的磷酸二酯酶 (PDE) 抑制剂，腺苷受体拮抗剂，和组蛋白脱乙酰酶 (HDAC) 活化剂。Theophylline (1,3-Dimethylxanthine) 抑制 PDE3 活性，放松气道平滑肌。Theophylline (1,3-Dimethylxanthine) 通过增加 IL-10 和抑制 NF-κ B进入细胞核而具有抗炎活性。Theophylline (1,3-Dimethylxanthine) 诱发细胞凋亡 (apoptosis)。Theophylline (1,3-Dimethylxanthine) 可用于哮喘和慢性阻塞性肺疾病 (COPD) 的研究。

熔点：271-273℃

沸点：454.1℃ at 760 mmHg

外观：白色至灰白色结晶粉末

溶解性：DMSO  :  11.11  mg/mL  (61.67  mM;  Need  ultrasonic)
H2O  :  5  mg/mL  (27.75  mM;  Need  ultrasonic)。

敏感性：对空气敏感

储存条件：2-8℃

注意：部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。

参考文献(31篇)

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